SCHEMBL8745248

SCHEMBL8745248

CCCCCC1CCC(C2CCC(CCC=Cc3ccc(OC(F)(F)F)cc3)CC2)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.35
GRIK2 Q13002 1/20 0.35
KDM1A O60341 1/20 0.35
RCOR1 Q9UKL0 1/20 0.35
EPHX2 P34913 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
LIPE Q05469 2/20 0.34
KDM2B Q8NHM5 1/20 0.34
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
CHRM4 P08173 1/20 0.33
TNNC1 P63316 1/20 0.33
BCHE P06276 2/20 0.32
ACHE P22303 2/20 0.32
BACE1 P56817 2/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745269 0.96 GRIK1 (0.37) GRIK1GRIK2KDM1ARCOR1EPHX2
SCHEMBL9137050 0.92 GRIK1 (0.37) GRIK1GRIK2KDM1ARCOR1EPHX2
SCHEMBL9139133 0.89 GRIK1 (0.37) GRIK1GRIK2KDM1ARCOR1EPHX2
SCHEMBL8745246 0.88 GRIK1 (0.39) GRIK1GRIK2KDM1ARCOR1HRH3
SCHEMBL8745294 0.85 GRIK1 (0.39) GRIK1GRIK2KDM1ARCOR1HRH3
SCHEMBL8745225 0.84 LSS (0.37) TNNC1
SCHEMBL8745282 0.84 TNNC1 (0.41) TNNC1
SCHEMBL8745261 0.84 TNNC1 (0.36) SLC6A4SLC6A3TNNC1
SCHEMBL9139977 0.84 EPHX2 (0.34) EPHX2
SCHEMBL9188507 0.83 AHR (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563981-B1 Cis-1,4-substituted 2-butene derivative CHISSO CORP (JP) 1997-01-22 EP disclosed
US-5401434-A Cis-1,4-substituted 2-butene derivative CHISSO CORPORATION (JP) 1995-03-28 US disclosed
EP-0563981-A2 Cis-1,4-substituted 2-butene derivative Chisso Corporation (JP) 1993-10-06 EP disclosed