SCHEMBL8745772

SCHEMBL8745772

COc1cc(OC)c2c(C)c(CCN3CCN(c4cccc(C(F)(F)F)c4)CC3)c(=O)oc2c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 2/20 0.51
ABCB1 P08183 4/20 0.49
ABCC1 P33527 2/20 0.49
SIGMAR1 Q99720 1/20 0.47
HTR1A P08908 2/20 0.47
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
HTR7 P34969 2/20 0.47
HTR6 P50406 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
BRAF P15056 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745755 0.88 ABCC1 (0.59) CCR4ABCB1ABCC1HTR1AHTR2A
SCHEMBL8745788 0.82 ABCC1 (0.56) CCR4ABCC1HTR1AHTR2AHTR7
SCHEMBL8745761 0.81 ABCC1 (0.54) CCR4ABCB1ABCC1HTR1AHTR2A
SCHEMBL8745799 0.81 ABCC1 (0.55) CCR4ABCB1ABCC1HTR1AHTR2A
SCHEMBL8745757 0.79 ABCC1 (0.54) CCR4ABCB1ABCC1HTR1AHTR2A
SCHEMBL8745763 0.78 ADRA1A (0.55) CCR4ABCC1HTR1AHTR2A
SCHEMBL8745802 0.76 ABCC1 (0.51) CCR4ABCB1ABCC1KDM4E
SCHEMBL11630455 0.76 TSHR (0.56) ABCB1SIGMAR1HTR1AHTR2AHTR2C
SCHEMBL8745779 0.75 NPSR1 (0.50) ABCC1HTR1AHTR2AHTR2CTSHR
SCHEMBL8745807 0.74 ABCC1 (0.49) CCR4ABCB1ABCC1SIGMAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663911-B1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE SCHWABE WILLMAR GMBH & CO (DE) 1997-02-05 EP disclosed
US-5550129-A THERAPY FOR NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS WILLMAR SCHWABE GMBH & CO. (DE) 1996-08-27 US disclosed