SCHEMBL8745757

SCHEMBL8745757

COc1cc(OC)c2c(C)c(CCN3CCN(c4ccccc4O)CC3)c(=O)oc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 2/20 0.54
CCR4 P51679 2/20 0.52
TP53 P04637 1/20 0.49
ABCB1 P08183 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
ADRA1A P35348 1/20 0.43
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745788 0.92 ABCC1 (0.56) ABCC1CCR4TP53GAAHTR1A
SCHEMBL8745799 0.91 ABCC1 (0.55) ABCC1CCR4TP53ABCB1ABCG2
SCHEMBL8745761 0.89 ABCC1 (0.54) ABCC1CCR4TP53ABCB1ABCG2
SCHEMBL8745763 0.88 ADRA1A (0.55) ABCC1CCR4TP53HTR1ADRD2
SCHEMBL8745755 0.87 ABCC1 (0.59) ABCC1CCR4TP53ABCB1ABCG2
SCHEMBL8745817 0.83 CCR4 (0.54) CCR4KDM4EALDH1A1GAAMAPT
SCHEMBL8745781 0.82 ADRA1A (0.51) ABCC1HTR1ADRD2HTR2AADRA1A
SCHEMBL8745808 0.81 DRD2 (0.52) HTR1ADRD2HTR2AADRA1AKCNH2
SCHEMBL8745807 0.80 ABCC1 (0.49) ABCC1CCR4TP53ABCB1ABCG2
SCHEMBL8745802 0.80 ABCC1 (0.51) ABCC1CCR4TP53ABCB1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663911-B1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE SCHWABE WILLMAR GMBH & CO (DE) 1997-02-05 EP disclosed
US-5550129-A THERAPY FOR NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS WILLMAR SCHWABE GMBH & CO. (DE) 1996-08-27 US disclosed
EP-0663911-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE. SCHWABE WILLMAR GMBH & CO (DE) 1995-07-26 EP disclosed
WO-1994008985-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE DR. WILLMAR SCHWABE GMBH & CO. (DE) 1994-04-28 WO disclosed