SCHEMBL8745779

SCHEMBL8745779

COc1cc2oc(=O)c(CCN3CCN(c4ccccc4)CC3)c(C)c2c(OC)c1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
DRD2 P14416 3/20 0.49
NR1I2 O75469 1/20 0.49
ADRB1 P08588 1/20 0.49
HTR1A P08908 1/20 0.49
ADRA2A P08913 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
SLC6A2 P23975 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
PTGS2 P35354 1/20 0.49
HRH1 P35367 1/20 0.49
HTR2B P41595 1/20 0.49
CHRNA4 P43681 1/20 0.49
SLC6A3 Q01959 1/20 0.49
PDE4D Q08499 1/20 0.49
KCNH2 Q12809 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745755 0.86 ABCC1 (0.59) NPSR1TDP1DRD2NR1I2ADRB1
SCHEMBL8745759 0.85 DRD2 (0.59) DRD2NR1I2ADRB1HTR1AADRA2A
SCHEMBL8745803 0.85 APP (0.45) DRD3ALDH1A1TSHRPPARGNCOA2
SCHEMBL8745782 0.80 DRD2 (0.54) DRD2NR1I2ADRB1HTR1AADRA2A
SCHEMBL8745788 0.76 ABCC1 (0.56) DRD2HTR1AHTR2AKCNH2TP53
SCHEMBL8745799 0.76 ABCC1 (0.55) DRD2HTR1AHTR2AKCNH2TP53
SCHEMBL8809027 0.75 DRD2 (0.59) DRD2NR1I2ADRB1HTR1AADRA2A
SCHEMBL8745772 0.75 CCR4 (0.51) TDP1HTR1AHTR2AHTR2CTSHR
SCHEMBL8745817 0.75 CCR4 (0.54) DRD2HTR1ADRD3ALDH1A1MAPT
SCHEMBL8745798 0.74 BRAF (0.56) DRD2HTR1AHTR2AKCNH2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663911-B1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE SCHWABE WILLMAR GMBH & CO (DE) 1997-02-05 EP disclosed
US-5550129-A THERAPY FOR NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS WILLMAR SCHWABE GMBH & CO. (DE) 1996-08-27 US disclosed
EP-0663911-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE. SCHWABE WILLMAR GMBH & CO (DE) 1995-07-26 EP disclosed
WO-1994008985-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE DR. WILLMAR SCHWABE GMBH & CO. (DE) 1994-04-28 WO disclosed