SCHEMBL8745808

SCHEMBL8745808

CCCOc1cc(OCCC)c2c(C)c(CCN3CCN(c4ccccc4OC)CC3)c(=O)oc2c1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.52
HTR2A P28223 1/20 0.52
ADRA1A P35348 1/20 0.52
KCNH2 Q12809 1/20 0.51
HTR1A P08908 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745781 0.92 ADRA1A (0.51) DRD2HTR2AADRA1AKCNH2HTR1A
SCHEMBL8745788 0.89 ABCC1 (0.56) DRD2HTR2AADRA1AKCNH2HTR1A
SCHEMBL8745763 0.86 ADRA1A (0.55) DRD2HTR2AADRA1AKCNH2HTR1A
SCHEMBL9144743 0.85 DRD2 (0.51) DRD2HTR2AADRA1AKCNH2HTR1A
SCHEMBL8745799 0.83 ABCC1 (0.55) DRD2HTR2AADRA1AKCNH2HTR1A
SCHEMBL8745757 0.81 ABCC1 (0.54) DRD2HTR2AADRA1AKCNH2HTR1A
SCHEMBL8745761 0.81 ABCC1 (0.54) HTR2AHTR1A
SCHEMBL8745817 0.80 CCR4 (0.54) DRD2ADRA1AHTR1A
SCHEMBL8745809 0.80 HTR2A (0.60) DRD2HTR2AADRA1AKCNH2HTR1A
SCHEMBL8745755 0.79 ABCC1 (0.59) DRD2HTR2AKCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663911-B1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE SCHWABE WILLMAR GMBH & CO (DE) 1997-02-05 EP disclosed
US-5550129-A THERAPY FOR NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS WILLMAR SCHWABE GMBH & CO. (DE) 1996-08-27 US disclosed
EP-0663911-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE. SCHWABE WILLMAR GMBH & CO (DE) 1995-07-26 EP disclosed
WO-1994008985-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE DR. WILLMAR SCHWABE GMBH & CO. (DE) 1994-04-28 WO disclosed