SCHEMBL874643

SCHEMBL874643

CCn1cc(-c2ccc(N)cc2)cc1C(=O)NCCN1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 1/20 0.50
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
KMT2A Q03164 3/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALDH1A1 P00352 2/20 0.43
HSD17B10 Q99714 2/20 0.43
MEN1 O00255 2/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
HTR4 Q13639 1/20 0.43
GLA P06280 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874641 0.85 LMNA (0.49) CHRNB2CHRNB4CHRNA3CHRNA4KMT2A
SCHEMBL882909 0.79 NAMPT (0.49) KMT2AMEN1JAK2
SCHEMBL13659640 0.75 MEN1 (0.50) KMT2ANPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL3401326 0.74 CYP1A2 (0.74) CD274KMT2ANPSR1CYP1A2CYP2D6
SCHEMBL3408343 0.73 ALDH1A1 (0.71) CD274KMT2ANPSR1CYP1A2CYP2D6
SCHEMBL874264 0.70 ALDH1A1 (0.55) CD274KMT2ACYP1A2CYP2D6CYP2C9
SCHEMBL2524048 0.70 KDM4E (0.46) CD274KMT2ANPSR1ALDH1A1HSD17B10
SCHEMBL877527 0.69 IKBKB (0.44) CD274NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL14262463 0.68 NPSR1 (0.50) CHRNB2CHRNB4CHRNA3CHRNA4KMT2A
SCHEMBL1186358 0.68 HTR4 (0.69) ALDH1A1HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed