SCHEMBL8747258

SCHEMBL8747258

COc1cc2c(cc1OC)C(C1(c3ccccc3Br)CCC1)NCC2.O=C(O[C@@H](C(=O)O)[C@@H](OC(=O)c1ccccc1)C(=O)O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.44
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
TSHR P16473 2/20 0.36
TP53 P04637 1/20 0.36
DRD1 P21728 1/20 0.35
DRD5 P21918 1/20 0.35
MTNR1B P49286 1/20 0.35
MAOA P21397 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
PRMT5 O14744 1/20 0.34
EGFR P00533 1/20 0.34
SLC6A9 P48067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747148 0.86 PKM (0.55) PKMKMT2AMEN1TSHRDRD1
SCHEMBL8747254 0.85 PKM (0.46) PKMKMT2AMEN1TSHRDRD1
Hydrochloric Acid SCHEMBL8747055 0.70 PKM (0.54) PKMKMT2AMEN1TSHRMAOA
SCHEMBL8747147 0.69 PKM (0.46) PKMKMT2AMEN1SLC6A9
SCHEMBL8747203 0.68 PKM (0.47) PKMKMT2AMEN1TSHRDRD1
SCHEMBL8747215 0.68 PKM (0.54) PKMKMT2AMEN1TSHRMAOA
SCHEMBL8747118 0.68 PKM (0.54) PKMKMT2AMEN1TSHRMAOA
SCHEMBL8747329 0.68 PKM (0.45) PKMKMT2AMEN1
SCHEMBL8747282 0.67 SLC6A9 (0.51) PKMKMT2AMEN1TSHRMAOA
SCHEMBL8747173 0.67 MAOA (0.47) KMT2AMEN1DRD1DRD5MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed