SCHEMBL8747217

SCHEMBL8747217

COc1ccccc1C1(C(=O)Cl)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.44
KMT2A Q03164 1/20 0.43
HTT P42858 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
OPRL1 P41146 1/20 0.41
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
CA4 P22748 1/20 0.40
CHRM2 P08172 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8110630 0.95 SIGMAR1 (0.47) SIGMAR1L3MBTL1KMT2AHTTHDAC3
SCHEMBL1465128 0.84 SIGMAR1 (0.50) SIGMAR1L3MBTL1KMT2AHTTHDAC3
SCHEMBL3144864 0.83 SIGMAR1 (0.49) SIGMAR1L3MBTL1KMT2AHTTHDAC3
SCHEMBL10002496 0.83 LMNA (0.53) SIGMAR1L3MBTL1KMT2AHTTHDAC3
SCHEMBL21034824 0.81 SIGMAR1 (0.47) SIGMAR1L3MBTL1KMT2AHTTHDAC3
SCHEMBL30038985 0.81 SIGMAR1 (0.47) SIGMAR1L3MBTL1KMT2AHTTHDAC3
SCHEMBL7464907 0.79 L3MBTL1 (0.55) SIGMAR1L3MBTL1KMT2AHTTHDAC3
SCHEMBL3443849 0.79 L3MBTL1 (0.51) SIGMAR1L3MBTL1KMT2AHTTHDAC3
SCHEMBL30683848 0.78 L3MBTL1 (0.54) SIGMAR1L3MBTL1KMT2AHTTHDAC3
SCHEMBL7457587 0.78 L3MBTL1 (0.54) SIGMAR1L3MBTL1KMT2AHTTHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed