SCHEMBL8747263

SCHEMBL8747263

COc1cccc(C(Cl)C#N)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
ACHE P22303 1/20 0.42
CASR P41180 4/20 0.42
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
KMT2A Q03164 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
NAAA Q02083 1/20 0.40
PGR P06401 1/20 0.40
AR P10275 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17466002 0.81 ALDH1A1 (0.48) AOC3L3MBTL1ACHECASRCES2
SCHEMBL4716539 0.81 ALDH1A1 (0.46) ALDH1A1CYP3A4PDE4APDE4BPDE4C
SCHEMBL10905926 0.81 PTGS1 (0.49) KMT2AALDH1A1
SCHEMBL954319 0.80 CASR (0.46) AOC3L3MBTL1ACHECASRCES2
SCHEMBL5263393 0.79 AOC3 (0.50) AOC3L3MBTL1ACHECASRCES2
SCHEMBL1055834 0.79 AOC3 (0.55) AOC3L3MBTL1ACHECES2CES1
SCHEMBL28782471 0.79 KMT2A (0.45) AOC3L3MBTL1ACHECASRCES2
SCHEMBL15775360 0.79 AOC3 (0.47) AOC3L3MBTL1ACHECASRCES2
SCHEMBL29066017 0.79 AOC3 (0.46) AOC3L3MBTL1ACHECASRCES2
SCHEMBL29175442 0.79 TRPA1 (0.52) AOC3L3MBTL1ACHECASRCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618900-B1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS KNOLL AG (DE) 1997-03-12 EP disclosed
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed