SCHEMBL874728

SCHEMBL874728

O=C(O)c1cc(-c2ccc([N+](=O)[O-])cc2)n[nH]1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.72
ALPL P05186 10/20 0.65
CA12 O43570 5/20 0.65
TP53 P04637 1/20 0.64
RPA1 P27694 1/20 0.63
CA9 Q16790 3/20 0.58
MAPT P10636 3/20 0.56
MEN1 O00255 1/20 0.56
NPC1 O15118 1/20 0.56
POLB P06746 1/20 0.56
PKM P14618 1/20 0.56
RAB9A P51151 1/20 0.56
KMT2A Q03164 1/20 0.56
MCL1 Q07820 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
MARS1 P56192 1/20 0.53
KDM4E B2RXH2 1/20 0.51
CACNA1B Q00975 1/20 0.47
APBA1 Q02410 1/20 0.47
PTPN1 P18031 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29444429 0.87 SMN1; SMN2 (0.56) SMN1; SMN2ALPLCA12TP53RPA1
SCHEMBL29196676 0.83 MAPT (0.68) SMN1; SMN2ALPLCA9MAPTMEN1
SCHEMBL22327632 0.80 SMN1; SMN2 (0.58) SMN1; SMN2TP53MAPTMEN1NPC1
SCHEMBL9267835 0.80 MAPT (0.60) SMN1; SMN2ALPLCA12MAPTMEN1
SCHEMBL1414100 0.79 ALPL (1.00) SMN1; SMN2ALPLCA12TP53RPA1
SCHEMBL726574 0.79 TP53 (1.00) SMN1; SMN2ALPLCA12TP53RPA1
SCHEMBL12490766 0.78 RAB9A (0.85) MAPTMEN1NPC1POLBPKM
SCHEMBL23803931 0.78 ALPL (0.73) SMN1; SMN2ALPLCA12TP53RPA1
SCHEMBL3447352 0.78 ALPL (1.00) ALPLCA12TP53RPA1CA9
SCHEMBL645330 0.78 ALPL (1.00) ALPLCA12TP53RPA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117886821-A Nitrogen-containing condensed ring derivative inhibitor, preparation method and application thereof 江苏豪森药业集团有限公司 2024-04-16 CN disclosed
CN-113754587-B Phenylpyrazole compound and application thereof 沈阳药科大学 2023-07-14 CN disclosed
CN-113754587-A Phenylpyrazole compound and application thereof 沈阳药科大学 2021-12-07 CN disclosed
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed