SCHEMBL874730

SCHEMBL874730

Nc1ccc(-c2nc(C(F)(F)C(F)(F)F)c(C(=O)NC3CC3)s2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 1/20 0.39
HDAC4 P56524 1/20 0.38
KDM4E B2RXH2 2/20 0.38
CHRM4 P08173 2/20 0.38
GRM1 Q13255 1/20 0.37
RAB9A P51151 5/20 0.37
MAPT P10636 2/20 0.37
MAPK11 Q15759 1/20 0.37
MAPK14 Q16539 1/20 0.37
CYP3A4 P08684 1/20 0.37
HTR2B P41595 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
SMYD3 Q9H7B4 1/20 0.36
TP53 P04637 2/20 0.36
MDM2 Q00987 2/20 0.36
ACVR2A P27037 1/20 0.36
TGFBR2 P37173 1/20 0.36
PPARA Q07869 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874117 0.80 RAB9A (0.48) NPC1ALDH1A1GAAKDM4ERAB9A
SCHEMBL874231 0.77 CHRNA7 (0.43) NPC1ALDH1A1GAAKDM4ERAB9A
SCHEMBL874429 0.75 CDC7 (0.42) NPC1ALDH1A1KDM4ECHRM4GRM1
SCHEMBL882714 0.74 MAPT (0.57) ALDH1A1KDM4EMAPT
SCHEMBL874665 0.73 GAA (0.52) NPC1ALDH1A1GAAKDM4ERAB9A
SCHEMBL875382 0.71 NPC1 (0.40) NPC1ALDH1A1KDM4ECHRM4RAB9A
SCHEMBL24303241 0.71 NPC1 (0.52) NPC1ALDH1A1GAAHDAC4KDM4E
SCHEMBL873941 0.70 RAB9A (0.48) NPC1ALDH1A1GAAKDM4ERAB9A
SCHEMBL3402398 0.68 NPC1 (0.62) NPC1ALDH1A1GAAHDAC4CHRM4
SCHEMBL3633642 0.66 RAB9A (0.72) NPC1HDAC4RAB9AMAPTMAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed