SCHEMBL874429

SCHEMBL874429

Nc1ccc(-c2nc(-c3ccsc3)c(C(=O)NC3CC3)s2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 4/20 0.42
DBF4 Q9UBU7 4/20 0.42
DRD2 P14416 4/20 0.39
DRD4 P21917 4/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
CHRM4 P08173 1/20 0.38
GRM1 Q13255 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
MAPK14 Q16539 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
MAPT P10636 2/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
MAPK11 Q15759 1/20 0.37
CYP3A4 P08684 1/20 0.37
HTR2B P41595 1/20 0.37
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874741 0.85 KMT2A (0.48) CDC7DBF4DRD4ALDH1A1RAB9A
SCHEMBL874757 0.79 HDAC1 (0.44)
SCHEMBL874730 0.75 NPC1 (0.39) ALDH1A1KDM4ECHRM4GRM1MAPK14
SCHEMBL874800 0.66 RAB9A (0.62) CDC7DBF4ALDH1A1KDM4EHTT
SCHEMBL3633642 0.66 RAB9A (0.72) MAPK14NPC1RAB9AMAPTMAPK11
SCHEMBL18458070 0.65 IDH2 (0.53) DRD2DRD4ALDH1A1LMNAMAPK14
SCHEMBL28750952 0.65 GSK3B (0.51) CDC7DBF4ALDH1A1KDM4ELMNA
SCHEMBL9911636 0.64 MLLT1 (0.63) ALDH1A1LMNANPC1RAB9ATP53
SCHEMBL15296751 0.64 HDAC1 (0.58) DRD2ALDH1A1LMNANPC1RAB9A
SCHEMBL3442327 0.63 RAB9A (0.62) LMNAMAPK14NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed