SCHEMBL8747780

SCHEMBL8747780

COC12CCC(c3cccc(CBr)c3)(CC1)CC2

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.34
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
TRPA1 O75762 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
OPRM1 P35372 2/20 0.31
OPRL1 P41146 2/20 0.31
PNMT P11086 1/20 0.31
KDM1A O60341 1/20 0.30
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8747881 0.78 HDAC4 (0.40) OPRM1OPRL1PNMTHSD11B1
SCHEMBL9302960 0.76 ALOX5 (0.52) ALOX5
SCHEMBL9247121 0.75 SLC16A3 (0.46)
SCHEMBL27693324 0.74 OPRD1 (0.41) ALOX5CYP4F2CYP4A11TRPA1ALDH1A1
SCHEMBL1193890 0.74 ALOX5 (0.60) ALOX5
SCHEMBL22070497 0.71 CYP4F2 (0.43) CYP4F2CYP4A11OPRM1HSD11B1
SCHEMBL12185113 0.70 OPRL1 (0.42) ALOX5CYP4F2CYP4A11TRPA1ALDH1A1
Methoxymethane SCHEMBL28161427 0.70 TSHR (0.50) CYP4F2CYP4A11TRPA1ALDH1A1TSHR
SCHEMBL8747855 0.68
SCHEMBL8747861 0.68 IDO1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0599732-B1 Derivatives of 1-phenylbicyclo-2,2,2-octane, their preparation process and pharmaceutical compositions containing them ADIR (FR) 1997-03-12 EP disclosed
US-5403953-A Antiarthritic and -inflammatory agents ADIR ET COMPAGNIE (FR) 1995-04-04 US disclosed
EP-0599732-A1 Derivatives of 1-phenylbicyclo-2,2,2-octane, their preparation process and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-06-01 EP disclosed