SCHEMBL8750700

SCHEMBL8750700

O=C(O)Cc1ccccc1Cn1c(=O)[nH]c2nc[nH]c2c1=O

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 9/20 0.59
ADORA3 P0DMS8 8/20 0.59
PDE4A P27815 5/20 0.53
PDE4B Q07343 5/20 0.53
PDE4C Q08493 5/20 0.53
PDE4D Q08499 5/20 0.53
ADORA2A P29274 4/20 0.53
PNP P00491 1/20 0.43
TLR7 Q9NYK1 1/20 0.41
KMT2A Q03164 1/20 0.40
MPO P05164 1/20 0.40
TPO P07202 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6360066 0.82 ADORA2B (0.75) ADORA2BADORA3PDE4APDE4BPDE4C
SCHEMBL985620 0.77 ADORA2B (0.63) ADORA2BADORA3PDE4APDE4BPDE4C
SCHEMBL31060278 0.75 ADORA2B (1.00) ADORA2BADORA3PDE4APDE4BPDE4C
SCHEMBL9750957 0.74 ADORA2B (0.69) ADORA2BADORA3PDE4APDE4BPDE4C
SCHEMBL7326382 0.71 PDE4A (0.68) ADORA2BADORA3PDE4APDE4BPDE4C
SCHEMBL4014471 0.71 ADORA2A (0.63) ADORA2BADORA3PDE4APDE4BPDE4C
SCHEMBL4602969 0.71 ADORA2B (0.73) ADORA2BADORA3PDE4APDE4BPDE4C
SCHEMBL5677075 0.71 ADORA2B (0.62) ADORA2BADORA3PDE4APDE4BPDE4C
SCHEMBL13735421 0.70 ADORA2B (0.55) ADORA2BADORA3PDE4APDE4BPDE4C
SCHEMBL5515444 0.70 ADORA2A (0.71) ADORA2BADORA3PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0764647-A1 Substituted xanthins BAYER AG (DE) 1997-03-26 EP disclosed