SCHEMBL8750774

SCHEMBL8750774

CCCCNc1cncc(C#N)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.46
CHRNA4 P43681 1/20 0.46
ABCB1 P08183 2/20 0.41
ABCG2 Q9UNQ0 2/20 0.41
POLB P06746 1/20 0.37
KDM6B O15054 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
MGLL Q99685 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
TLR8 Q9NR97 3/20 0.34
TLR7 Q9NYK1 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
RAF1 P04049 1/20 0.33
ABCC1 P33527 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8750751 0.83 CHEK1 (0.42) CYP11B1CYP11B2RAF1
SCHEMBL14155105 0.75 TLR8 (0.47) ABCB1ABCG2TLR8TLR7ALDH1A1
SCHEMBL1419851 0.75 CHRNB2 (0.43) CHRNB2CHRNA4POLBKDM6BKDM4C
SCHEMBL8176730 0.74 ABCB1 (0.52) ABCB1ABCG2MGLLTLR8TLR7
SCHEMBL14007397 0.73 ALDH1A1 (0.44) CHRNB2CHRNA4CYP11B1CYP11B2KDM4E
SCHEMBL8244430 0.73 SCN10A (0.37) CHRNB2CHRNA4CYP11B1CYP11B2RAF1
SCHEMBL7220029 0.71 TSHR (0.44) CHRNB2CHRNA4ALDH1A1HPGDRAF1
SCHEMBL28133362 0.71 ABL1 (0.44) ABCB1ABCG2TLR8TLR7ALDH1A1
SCHEMBL18386511 0.70 ABL1 (0.43) CHRNB2CHRNA4
SCHEMBL8237778 0.70 KCNH2 (0.46) POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0634400-B1 PYRIDINECARBOXIMIDAMIDE COMPOUND AND USE THEREOF KIRIN BREWERY (JP) 1997-04-02 EP disclosed
US-5508293-A TREATING HYPERTENSION, ANGINA PECTORIS KIRIN BEER KABUSHIKI KAISHA (JP) 1996-04-16 US disclosed
EP-0634400-A1 PYRIDINECARBOXIMIDAMIDE COMPOUND AND USE THEREOF KIRIN BEER KABUSHIKI KAISHA (JP) 1995-01-18 EP disclosed