SCHEMBL8759775

SCHEMBL8759775

O=CC(Cl)N1CCN(C2COC(Cc3ccccc3)CO2)CC1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.32
DHFR P00374 1/20 0.32
KCNH2 Q12809 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
CCR3 P51677 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691572 0.75 GRM2 (0.35) GRM2
SCHEMBL6609808 0.75 SIGMAR1 (0.41) GRM2
SCHEMBL2688223 0.74 GRIN2B (0.55) GRM2
Hydrochloric Acid SCHEMBL9466555 0.74 SIGMAR1 (0.41) GRM2
SCHEMBL8303444 0.72 SIGMAR1 (0.55) CCR3
SCHEMBL6806817 0.72 CCR3 (0.55) KCNH2HRH3CCR3
SCHEMBL9179381 0.71 ALDH1A1 (0.40)
SCHEMBL9179397 0.71 SIGMAR1 (0.55)
SCHEMBL9173695 0.70 ALDH1A1 (0.37) HRH3
SCHEMBL9178363 0.69 SIGMAR1 (0.41) CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773937-A1 NOVEL ARYL PIPERAZINE-DERIVED PIPERAZIDE DERIVATIVES, METHODS FOR THEIR PREPARATION, THEIR USE AS DRUGS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME PIERRE FABRE MEDICAMENT (FR) 1997-05-21 EP disclosed
WO-1996002525-A1 NOVEL ARYL PIPERAZINE-DERIVED PIPERAZIDE DERIVATIVES, METHODS FOR THEIR PREPARATION, THEIR USE AS DRUGS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME PIERRE FABRE MEDICAMENT (FR) 1996-02-01 WO disclosed