SCHEMBL876171

SCHEMBL876171

CN(C(=O)c1ccc2c(c1)C(N1C=C(C(=O)O)C=NC1)CC2(C)C)C1CCN(c2ccncc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
ALOX15 P16050 1/20 0.36
CCR5 P51681 1/20 0.35
F10 P00742 4/20 0.34
HRH3 Q9Y5N1 2/20 0.32
JAK2 O60674 5/20 0.32
JAK1 P23458 5/20 0.32
POLB P06746 1/20 0.32
USP2 O75604 1/20 0.31
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31
PDK2 Q15119 1/20 0.30
ROCK2 O75116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878507 0.87 CCR5 (0.35) CCR5F10JAK2JAK1POLB
SCHEMBL876130 0.86 POLB (0.35) CCR5F10JAK2JAK1POLB
SCHEMBL875757 0.84 CCR5 (0.35) CCR5F10JAK2JAK1POLB
SCHEMBL876267 0.84 F10 (0.36) CCR5F10JAK2JAK1POLB
SCHEMBL875502 0.79 ALDH1A1 (0.34) ALDH1A1ALOX15CCR5F10POLB
SCHEMBL786192 0.79 ALDH1A1 (0.46) ALDH1A1ALOX15CCR5F10HRH3
SCHEMBL785791 0.76 ALDH1A1 (0.41) ALDH1A1ALOX15CCR5F10JAK2
SCHEMBL784500 0.74 ALDH1A1 (0.39) ALDH1A1ALOX15CCR5F10JAK2
SCHEMBL784256 0.74 CCR5 (0.38) ALDH1A1ALOX15CCR5F10HRH3
SCHEMBL784953 0.73 POLB (0.39) ALDH1A1ALOX15CCR5F10POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed