SCHEMBL876267

SCHEMBL876267

CN(C(=O)c1ccc2c(c1)C(N1C=C(C(=O)O)C=NC1)CCO2)C1CCN(c2ccncc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F10 P00742 4/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
CCR5 P51681 1/20 0.34
KDM4C Q9H3R0 3/20 0.33
KDM6B O15054 1/20 0.33
GPR55 Q9Y2T6 1/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
POLB P06746 1/20 0.31
USP2 O75604 1/20 0.31
ROCK2 O75116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878507 0.87 CCR5 (0.35) F10CCR5KDM4CGPR55JAK2
SCHEMBL876130 0.85 POLB (0.35) F10CCR5KDM4CKDM6BGPR55
SCHEMBL875757 0.85 CCR5 (0.35) F10CCR5KDM4CGPR55JAK2
SCHEMBL876171 0.84 ALDH1A1 (0.36) F10CCR5JAK2JAK1POLB
SCHEMBL876159 0.79 NPC1 (0.35) F10NPC1RAB9ACCR5KDM4C
SCHEMBL784870 0.79 F10 (0.42) F10NPC1RAB9ACCR5POLB
SCHEMBL876268 0.78 F10 (0.34) F10NPC1RAB9ACCR5KDM4C
SCHEMBL876160 0.78 F10 (0.33) F10NPC1RAB9ACCR5
SCHEMBL784756 0.76 F10 (0.40) F10NPC1RAB9ACCR5KDM4C
SCHEMBL785183 0.75 F10 (0.39) F10NPC1RAB9ACCR5POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed