SCHEMBL8763135

SCHEMBL8763135

CCC(CCc1ccncc1)(NC(C)=O)C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
ALDH1A1 P00352 1/20 0.38
RAB9A P51151 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.35
HTT P42858 1/20 0.35
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NAMPT P43490 1/20 0.34
KDR P35968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29842432 0.73 PKM (0.35) HTT
SCHEMBL16892930 0.72 LOXL2 (0.47) ALDH1A1RAB9ASMN1; SMN2NPC1LOXL2
SCHEMBL4406979 0.71 ALDH1A1 (0.38) ALDH1A1RAB9ANPC1
SCHEMBL13811853 0.70 MAOA (0.42) ALDH1A1RAB9ANPC1
SCHEMBL12733180 0.69 ALDH1A1 (0.59) TSHRALDH1A1SMN1; SMN2HTT
SCHEMBL13821633 0.68 ALDH1A1 (0.38) ALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL6501640 0.66 ACACB (0.49) TSHRALDH1A1RAB9AHTT
SCHEMBL424305 0.65 KDM4E (0.65) TSHRALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL14889554 0.65 LOXL2 (0.47) TSHRALDH1A1RAB9ASMN1; SMN2NPC1
SCHEMBL28773068 0.65 BLM (0.45) ALDH1A1RAB9ASMN1; SMN2NPC1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636141-B1 PYRIMIDINYL ACETAMIDES AS ELASTASE INHIBITORS ZENECA LTD (GB) 1997-06-25 EP disclosed