SCHEMBL8763146

SCHEMBL8763146

CCCCOC(=O)N1CC(Oc2ccccc2)CC1C(=O)OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.41
ECE1 P42892 1/20 0.40
MCL1 Q07820 5/20 0.40
HRH3 Q9Y5N1 2/20 0.40
MMP2 P08253 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPK1 P28482 1/20 0.39
KCNH2 Q12809 1/20 0.39
NPFFR1 Q9GZQ6 1/20 0.38
NPFFR2 Q9Y5X5 1/20 0.38
BCHE P06276 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
HPGD P15428 1/20 0.38
ATM Q13315 1/20 0.38
P2RY12 Q9H244 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8763150 1.00 P2RX3 (0.41) P2RX3ECE1MCL1HRH3MMP2
SCHEMBL7015458 0.84 POLB (0.47) MCL1KDM4E
SCHEMBL2298566 0.84 POLB (0.47) MCL1KDM4E
SCHEMBL7015459 0.84 POLB (0.47) MCL1KDM4E
SCHEMBL28233898 0.82 GBA2 (0.40) P2RX3ECE1MMP2L3MBTL1KDM4E
SCHEMBL7020775 0.82 ALDH1A1 (0.48) MCL1MMP2KDM4E
SCHEMBL7020805 0.82 ALDH1A1 (0.48) MCL1MMP2KDM4E
SCHEMBL15719248 0.81 MMP2 (0.47) P2RX3HRH3MMP2KCNH2
SCHEMBL13758532 0.81 ALDH1A1 (0.46) L3MBTL1KDM4EMAPK1
SCHEMBL15719188 0.80 P2RX3 (0.51) P2RX3MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784628-A1 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1997-07-23 EP disclosed
WO-1995035308-A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-12-28 WO disclosed