SCHEMBL8764666

SCHEMBL8764666

CC(C)CCC(=N)NCCCN1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.45
TP53 P04637 2/20 0.45
FPR3 P25089 1/20 0.42
FPR2 P25090 1/20 0.42
RAD52 P43351 1/20 0.38
TSHR P16473 2/20 0.38
CYP1A2 P05177 2/20 0.38
USP2 O75604 1/20 0.38
MAPK1 P28482 1/20 0.38
HRH3 Q9Y5N1 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ATM Q13315 1/20 0.36
HTR4 Q13639 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8763757 0.95 FPR3 (0.46) SMN1; SMN2TP53FPR3FPR2RAD52
SCHEMBL8971745 0.76 FPR3 (0.36) SMN1; SMN2TP53FPR3FPR2RAD52
Hydrochloric Acid SCHEMBL8972332 0.75 RAD52 (0.37) SMN1; SMN2TP53FPR3FPR2RAD52
Hydrochloric Acid SCHEMBL6584702 0.75 FPR3 (0.52) SMN1; SMN2TP53FPR3FPR2RAD52
SCHEMBL9329964 0.74 SCN5A (0.50) SMN1; SMN2TP53FPR3FPR2HRH3
SCHEMBL20363769 0.73 L3MBTL1 (0.44) SMN1; SMN2TP53MAPK1HRH3ALDH1A1
SCHEMBL17525451 0.73 HRH3 (0.46) SMN1; SMN2TP53TSHRHRH3ALDH1A1
Hydrochloric Acid SCHEMBL9322363 0.72 SCN5A (0.49) SMN1; SMN2TP53FPR3FPR2RAD52
SCHEMBL172955 0.72 HRH3 (0.56) SMN1; SMN2CYP1A2MAPK1HRH3MEN1
SCHEMBL439729 0.72 HRH3 (0.56) SMN1; SMN2CYP1A2MAPK1HRH3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420116-B1 Novel substituted alkyl piperidines and their use as inhibitors of cholesterol synthesis MERRELL PHARMA INC (US) 1997-07-30 EP claimed
US-5217979-A Substituted alkyl piperidines MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-08 US claimed
EP-0420116-A2 Novel substituted alkyl piperidines and their use as inhibitors of cholesterol synthesis MERRELL PHARMACEUTICALS INC. (US) 1991-04-03 EP claimed
EP-0420116-B1 Novel substituted alkyl piperidines and their use as inhibitors of cholesterol synthesis MERRELL PHARMA INC (US) 1997-07-30 EP disclosed
US-5217979-A Substituted alkyl piperidines MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-08 US disclosed
EP-0420116-A2 Novel substituted alkyl piperidines and their use as inhibitors of cholesterol synthesis MERRELL PHARMACEUTICALS INC. (US) 1991-04-03 EP disclosed