SCHEMBL6999564

SCHEMBL6999564

O=C(O)C(C(=O)O)c1ncccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.44
PTPRA P18433 1/20 0.39
NAPRT Q6XQN6 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 2/20 0.39
P4HTM Q9NXG6 1/20 0.39
KDM4E B2RXH2 4/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
CYP3A4 P08684 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
BLM P54132 1/20 0.37
AGER Q15109 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8831554 0.75 PTGS2 (0.42) PTPRANAPRTL3MBTL1LMNAP4HTM
SCHEMBL9373154 0.74 SRC (0.41) SRCLMNAKDM4ETDP1ALDH1A1
Hydrochloric Acid SCHEMBL22775404 0.73 PTGS2 (0.41) PTPRANAPRTL3MBTL1LMNAP4HTM
SCHEMBL2647026 0.72 ALDH1A1 (0.50) L3MBTL1ALDH1A1ALOX15TSHRNPSR1
SCHEMBL3767996 0.72 SLC6A3 (0.52) SRCPTPRANAPRTL3MBTL1LMNA
SCHEMBL27940696 0.70 SRC (0.40) SRCPTPRANAPRTL3MBTL1LMNA
SCHEMBL24327756 0.70 KMT2A (0.35) PTPRANAPRTL3MBTL1LMNAP4HTM
SCHEMBL895966 0.70 LMNA (0.40) PTPRALMNAKDM4EALDH1A1SMN1; SMN2
SCHEMBL8765939 0.70 CES2 (0.34) PTPRANAPRTL3MBTL1LMNAP4HTM
SCHEMBL26940504 0.70 KMT2A (0.35) PTPRANAPRTL3MBTL1LMNAP4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915875-B1 SUBSTITUTED TRIAZOLO-PYRIDAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME (GB) 2003-04-09 EP disclosed
US-6255305-B1 PSYCHOLOGICAL DISORDERS MERCK SHARP & DOHME LIMITED (GB) 2001-07-03 US disclosed