SCHEMBL8766530

SCHEMBL8766530

C#CC(CCCc1cccnn1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
CTDSP1 Q9GZU7 1/20 0.37
VNN1 O95497 2/20 0.36
CES1 P23141 1/20 0.35
CYP2C9 P11712 1/20 0.33
NAMPT P43490 1/20 0.33
P2RX7 Q99572 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PTPRA P18433 1/20 0.32
TBXAS1 P24557 1/20 0.31
NOS1 P29475 1/20 0.30
GLS O94925 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765876 0.76 NAAA (0.35) PTPRANOS1
SCHEMBL8766796 0.74 KDM4E (0.34) CYP1A2VNN1CYP2C9NAMPTTBXAS1
SCHEMBL6046250 0.73 CYP1A2 (0.50) CYP1A2CTDSP1VNN1CES1CYP2C19
SCHEMBL5326890 0.73 CYP1A2 (0.71) CYP1A2CTDSP1VNN1P2RX7NOS1
SCHEMBL27449978 0.72 TBXAS1 (0.53) CYP1A2CTDSP1CES1SMN1; SMN2TBXAS1
SCHEMBL18854185 0.72 CYP1A2 (0.44) CYP1A2CTDSP1VNN1CES1CYP2C9
SCHEMBL20224951 0.72 CYP1A2 (0.40) CYP1A2CTDSP1VNN1P2RX7CYP2C19
SCHEMBL9842898 0.71 TBXAS1 (0.54) CYP1A2CES1TBXAS1
SCHEMBL18110355 0.70 CYP1A2 (0.42) CYP1A2CTDSP1VNN1CES1CYP2C9
SCHEMBL2436110 0.70 CYP1A2 (0.50) CYP1A2CTDSP1VNN1CES1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1997-07-30 EP disclosed
WO-1996011686-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-04-25 WO disclosed