SCHEMBL8765876

SCHEMBL8765876

C#CC(CCCc1ncccn1)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.35
PTPRA P18433 1/20 0.32
IL1RN P18510 1/20 0.31
ERAP2 Q6P179 1/20 0.31
ERAP1 Q9NZ08 1/20 0.31
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766530 0.76 CYP1A2 (0.49) PTPRANOS1
SCHEMBL8766796 0.76 KDM4E (0.34) NOS1
SCHEMBL8765582 0.71 CYP2C19 (0.49)
SCHEMBL8766708 0.71 ALDH1A1 (0.49)
SCHEMBL15452338 0.70 MAPT (0.47)
SCHEMBL16672942 0.69 ERAP1 (0.46) IL1RNERAP2ERAP1
SCHEMBL2831370 0.69 TBXAS1 (0.47) NAAA
SCHEMBL1712974 0.67 LMNA (0.47)
SCHEMBL3936899 0.67 SMN1; SMN2 (0.52)
SCHEMBL5285402 0.67 ARG1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1997-07-30 EP disclosed
WO-1996011686-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-04-25 WO disclosed