SCHEMBL8766796

SCHEMBL8766796

C#CC(CCCc1cnccn1)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
NAPRT Q6XQN6 1/20 0.34
HCAR2 Q8TDS4 1/20 0.34
VNN1 O95497 2/20 0.34
LMNA P02545 2/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HPGD P15428 1/20 0.32
POLB P06746 1/20 0.31
TBXAS1 P24557 1/20 0.31
ABL1 P00519 1/20 0.31
RIN1 Q13671 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.30
NAMPT P43490 1/20 0.30
IDO1 P14902 1/20 0.30
NOS1 P29475 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765876 0.76 NAAA (0.35) NOS1
SCHEMBL8766530 0.74 CYP1A2 (0.49) VNN1TBXAS1CYP2C9NAMPTNOS1
SCHEMBL27486167 0.72 GNPAT (0.40) KDM4EVNN1LMNAMAPTPSMB11
SCHEMBL27734711 0.72 ADORA3 (0.40) KDM4ENAPRTHCAR2VNN1HDAC3
SCHEMBL27734710 0.72 ADORA3 (0.40) KDM4ENAPRTHCAR2VNN1HDAC3
SCHEMBL1649008 0.72 TBXAS1 (0.47) KDM4ENAPRTHCAR2VNN1HDAC3
SCHEMBL1648470 0.70 TBXAS1 (0.54) KDM4ENAPRTHCAR2TBXAS1MAPT
SCHEMBL28362525 0.70 HSP90AA1 (0.40) KDM4ENAPRTHCAR2VNN1HDAC3
SCHEMBL15798754 0.70 ALDH1A1 (0.36) KDM4EVNN1LMNAHDAC3HDAC1
SCHEMBL1648907 0.69 TBXAS1 (0.55) LMNATBXAS1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1997-07-30 EP disclosed
WO-1996011686-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-04-25 WO disclosed