SCHEMBL8767448

SCHEMBL8767448

COc1ccc2c(c1)C(C)(C)C(N)CC2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.54
DRD3 P35462 1/20 0.54
POLA1 P09884 4/20 0.53
CYP3A4 P08684 2/20 0.50
ALDH1A1 P00352 1/20 0.50
THRB P10828 1/20 0.50
MAPK1 P28482 1/20 0.50
KDM1A O60341 1/20 0.48
CYP2C9 P11712 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
ADRB2 P07550 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
SLC6A2 P23975 1/20 0.43
HTR2C P28335 1/20 0.43
HRH1 P35367 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRK1 P41145 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8768777 1.00 DRD2 (0.54) DRD2DRD3POLA1CYP3A4ALDH1A1
SCHEMBL3951310 0.89 KDM1A (0.57) DRD2DRD3POLA1CYP3A4ALDH1A1
SCHEMBL11290168 0.85 DRD2 (0.50) DRD2DRD3POLA1CYP3A4ALDH1A1
Hydrochloric Acid SCHEMBL11291604 0.83 DRD2 (0.49) DRD2DRD3POLA1CYP3A4ALDH1A1
SCHEMBL20366521 0.81 POLA1 (0.50) DRD2DRD3POLA1CYP3A4ALDH1A1
SCHEMBL1950165 0.78 OPRM1 (0.44) OPRM1OPRK1
SCHEMBL11297637 0.77 KDM1A (0.54) DRD2DRD3KDM1AADRB2HTR1A
Hydrochloric Acid SCHEMBL11296787 0.75 KDM1A (0.52) DRD2DRD3CYP3A4ALDH1A1KDM1A
SCHEMBL17988091 0.74 KDM1A (0.67) POLA1KDM1A
SCHEMBL5343873 0.74 KDM1A (0.50) MAPK1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0579833-B1 ETHANOLAMINE DERIVATIVES WITH ANTI-POLLAKIURIA ACTIVITY FUJISAWA PHARMACEUTICAL CO (JP) 1997-08-20 EP disclosed