SCHEMBL8768283

SCHEMBL8768283

COc1ccc2nc(SCCN(C)C)[nH]c2c1

nearest known ligand 0.97

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.97
CYP2E1 P05181 18/20 0.74
CYP2C8 P10632 18/20 0.74
CYP2D6 P10635 18/20 0.74
CYP2C9 P11712 18/20 0.74
CYP2B6 P20813 18/20 0.74
CYP2C19 P33261 18/20 0.74
CYP1A2 P05177 17/20 0.74
CYP3A4 P08684 16/20 0.74
BRS3 P32247 1/20 0.63
HRH4 Q9H3N8 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8768278 0.90 LMNA (0.79) LMNACYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL14304388 0.85 CYP2E1 (0.90) LMNACYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL10492884 0.82 HRH4 (0.70) LMNACYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL9743301 0.81 CYP2E1 (0.76) LMNACYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL22468990 0.81 CYP2E1 (1.00) LMNACYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL12963120 0.80 CYP1A2 (0.67) LMNACYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL17153978 0.78 CYP2E1 (0.72) LMNACYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL9512670 0.77 ALDH1A1 (0.83) LMNAHRH4
SCHEMBL7672276 0.77 CYP2E1 (0.70) LMNACYP2E1CYP2C8CYP2D6CYP2C9
SCHEMBL4650010 0.76 CYP2E1 (1.00) LMNACYP2E1CYP2C8CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0788795-A1 PHARMACOLOGICALLY ACTIVE 2-MERCAPTOBENZIMIDAZOLE DERIVATIVES NAUCHNO-ISSLEDOVATELSKY INSTITUT FARMAKOLOGII AKADEMII MEDITSINSKIKH NAUK (RU) 1997-08-13 EP disclosed