SCHEMBL8769018

SCHEMBL8769018

N#Cc1ccccc1NC1=CCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
TSHR P16473 3/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41
GAA P10253 3/20 0.40
AURKA O14965 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 3/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
MEN1 O00255 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8984047 0.90 FLT1 (0.40) KDM4ETSHRHPGDHSD17B10FLT1
SCHEMBL30804592 0.80 KDM4E (0.55) KDM4ETSHRHPGDHSD17B10FLT1
SCHEMBL30804597 0.80 KDM4E (0.55) KDM4ETSHRHPGDHSD17B10FLT1
SCHEMBL395135 0.80 KDM4E (0.55) KDM4ETSHRHPGDHSD17B10FLT1
SCHEMBL9874246 0.76 TAS1R3 (0.41) KDM4ETSHRHPGDHSD17B10FLT1
SCHEMBL8984088 0.74 MT-CO2 (0.45) KDM4ETSHRHPGDHSD17B10FLT1
Hydrochloric Acid SCHEMBL9875354 0.73 MT-CO2 (0.44) KDM4ETSHRHPGDHSD17B10FLT1
SCHEMBL4188631 0.72 AURKA (0.59) KDM4ETSHRHPGDHSD17B10FLT1
SCHEMBL3286845 0.69 KDM4E (0.46) KDM4ETSHRHPGDHSD17B10FLT1
SCHEMBL22497632 0.69 KDM4E (0.50) KDM4ETSHRHPGDHSD17B10FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0789690-A1 N-ARYL AND N-HETEROARYL-1,2-DIAMINOCYCLOBUTENE-3,4-DIONES WITH SMOOTH MUSCLE RELAXING ACTIVITIES AMERICAN HOME PRODUCTS CORPORATION (US) 1997-08-20 EP disclosed
WO-1996014300-A1 N-ARYL AND N-HETEROARYL-1,2-DIAMINOCYCLOBUTENE-3,4-DIONES WITH SMOOTH MUSCLE RELAXING ACTIVITIES AMERICAN HOME PRODUCTS CORPORATION (US) 1996-05-17 WO disclosed