SCHEMBL8770223

SCHEMBL8770223

N#Cc1ccc(C(=O)N=C=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.53
CA1 P00915 2/20 0.53
GSK3B P49841 2/20 0.53
PARP15 Q460N3 1/20 0.44
PARP10 Q53GL7 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
ALDH1A1 P00352 2/20 0.42
MAPT P10636 1/20 0.42
CA12 O43570 1/20 0.41
CA3 P07451 1/20 0.41
CA6 P23280 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
NPC1 O15118 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
RAB9A P51151 1/20 0.40
P4HB P07237 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3393415 0.85 TP53 (0.36) CA2CA1GSK3BALDH1A1MAPT
SCHEMBL572208 0.82 CA2 (0.52) CA2CA1GSK3BPARP15PARP10
SCHEMBL3205731 0.75 CES2 (0.50) CA2CA1GSK3BALDH1A1MAPT
SCHEMBL811028 0.75 ALDH1A1 (0.50) GSK3BALDH1A1MAPTNPC1MEN1
SCHEMBL15540018 0.75 TPMT (0.48) CA2CA1GSK3BSLC6A3
SCHEMBL67959 0.75 CES2 (0.50) CA2CA1ALDH1A1MAPTNPC1
SCHEMBL28364182 0.75 MAPT (0.42) CA2CA1PARP10ALDH1A1MAPT
SCHEMBL4247526 0.75 CES2 (0.50) CA2CA1GSK3BMAPTCA12
SCHEMBL84542 0.74 CES1 (0.46) CA2CA1ALDH1A1MAPTCA12
SCHEMBL11139683 0.74 CES1 (0.46) CA2CA1ALDH1A1MAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632019-B1 Acylureas ZENECA LTD (GB) 1997-09-24 EP disclosed
US-5576334-A ANTICOAGULANTS ZENECA LIMITED (GB) 1996-11-19 US disclosed
EP-0632019-A1 Acylureas ZENECA LIMITED (GB) 1995-01-04 EP disclosed