SCHEMBL8771828

SCHEMBL8771828

CC(COc1ccc(Cl)cn1)NC(=O)[C@@H](NC(=O)Oc1ccccc1)C(C)C

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.45
MTNR1A P48039 3/20 0.42
MTNR1B P49286 3/20 0.42
TRPA1 O75762 1/20 0.41
SLC1A3 P43003 1/20 0.41
LIPE Q05469 1/20 0.41
CNR1 P21554 2/20 0.39
CNR2 P34972 1/20 0.39
RAB9A P51151 1/20 0.38
ACACB O00763 1/20 0.37
CYP1A2 P05177 1/20 0.37
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
CDK5 Q00535 1/20 0.36
MMP1 P03956 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8771843 0.85 TRPA1 (0.44) TRPA1CNR1CNR2ACACBMMP1
SCHEMBL9225370 0.85 LIPE (0.40) CCR1MTNR1AMTNR1BTRPA1LIPE
Hydrochloric Acid SCHEMBL8771984 0.76 MEN1 (0.41) TRPA1CNR1CNR2ACACBMMP1
SCHEMBL8771906 0.76 MTNR1A (0.50) MTNR1AMTNR1BSLC1A3
SCHEMBL8771836 0.75 MTNR1A (0.49) MTNR1AMTNR1BSLC1A3CYP1A2
SCHEMBL8771754 0.75 MTNR1A (0.49) MTNR1AMTNR1BSLC1A3ACACBCYP1A2
SCHEMBL8607199 0.74 TSHR (0.51) CCR1RAB9A
SCHEMBL8607205 0.74 TSHR (0.51) CCR1RAB9A
SCHEMBL9228363 0.72 MMP1 (0.40) TRPA1CNR1CNR2RAB9AACACB
Hydrochloric Acid SCHEMBL8771979 0.71 MMP1 (0.41) TRPA1CNR1CNR2ACACBMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0648740-B1 AMINO ACID AMIDE DERIVATIVE, AGROHORTICULTURAL BACTERICIDE, AND PRODUCTION PROCESS KUMIAI CHEMICAL INDUSTRY CO (JP) 1997-10-08 EP disclosed
EP-0648740-A1 AMINO ACID AMIDE DERIVATIVE, AGROHORTICULTURAL BACTERICIDE, AND PRODUCTION PROCESS KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1995-04-19 EP disclosed