Naphthalene

Naphthalene

SCHEMBL8773082

Cl.O=S(=O)(O)O.c1ccc2ccccc2c1

nearest known ligand 0.53

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Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Naphthalene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 2/20 0.53
CYP2A6 P11509 1/20 0.53
TSHR P16473 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
LMNA P02545 2/20 0.42
KDM4E B2RXH2 3/20 0.41
CA5A P35218 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
CA1 P00915 4/20 0.39
CA2 P00918 4/20 0.39
CA9 Q16790 3/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 1/20 0.39
CYP1A2 P05177 1/20 0.39
F2 P00734 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
PRSS3 P35030 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Naphthalene SCHEMBL2678900 0.97 ALOX12 (0.57) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL28674544 0.97 ALOX12 (0.57) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL5574575 0.97 ALOX12 (0.57) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL672294 0.97 ALOX12 (0.57) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL29361795 0.97 ALOX12 (0.57) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL28983768 0.93 ALOX12 (0.53) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL9484719 0.93 ALOX12 (0.53) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL9484717 0.93 ALOX12 (0.53) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL7145629 0.93 ALOX12 (0.53) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL28414009 0.90 ALOX12 (0.50) ALOX12CYP2A6TSHRSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0439585-B1 IMMOBILISATION OF LIGANDS BY RADIO-DERIVATIZED POLYMERS MAG GEORG MAYRHOFER & CO OHG (AT) 1997-10-29 EP disclosed
US-5196478-A Polystyrene, assays EPIPHARM ALLERGIE-SERVICE GESELLSCHAFT M.B.H. (AT) 1993-03-23 US disclosed
EP-0439585-A1 IMMOBILISATION OF LIGANDS BY RADIO-DERIVATIZED POLYMERS. EPIPHARM ALLERGIE SERVICE (AT) 1991-08-07 EP disclosed
WO-1991002768-A1 IMMOBILISATION OF LIGANDS BY RADIO-DERIVATIZED POLYMERS EPIPHARM ALLERGIE-SERVICE GESELLSCHAFT M.B.H. (AT) 1991-03-07 WO disclosed