Naphthalene

Naphthalene

SCHEMBL5574575

O=S(=O)(O)O.O=S(=O)(O)O.O=S(=O)(O)O.c1ccc2ccccc2c1

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Naphthalene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 2/20 0.57
CYP2A6 P11509 1/20 0.57
TSHR P16473 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
LMNA P02545 2/20 0.44
KDM4E B2RXH2 3/20 0.43
CA5A P35218 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
CYP1A2 P05177 1/20 0.41
CA1 P00915 4/20 0.41
CA2 P00918 4/20 0.41
CA9 Q16790 3/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 1/20 0.41
F2 P00734 1/20 0.40
PRSS1 P07477 1/20 0.40
PRSS2 P07478 1/20 0.40
PRSS3 P35030 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Naphthalene SCHEMBL28674544 1.00 ALOX12 (0.57) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL29361795 1.00 ALOX12 (0.57) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL2678900 1.00 ALOX12 (0.57) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL672294 1.00 ALOX12 (0.57) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL8773082 0.97 ALOX12 (0.53) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL9484717 0.97 ALOX12 (0.53) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL28983768 0.97 ALOX12 (0.53) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL9484719 0.97 ALOX12 (0.53) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL7145629 0.97 ALOX12 (0.53) ALOX12CYP2A6TSHRSMN1; SMN2LMNA
Naphthalene SCHEMBL1618294 0.94 ALOX12 (0.50) ALOX12CYP2A6TSHRSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070003987-A1 Screening method for substance binding to merozoite surface protein-1/42 MEDICAL RESEARCH COUNCIL (GB) 2007-01-04 US disclosed
EP-1634079-A1 SCREENING METHOD FOR SUBSTANCES BINDING TO MEROZOITE SURFACE PROTEIN-1/42 MEDICAL RESEARCH COUNCIL (GB) 2006-03-15 EP disclosed
WO-2004113920-A1 SCREENING METHOD FOR SUBSTANCES BINDING TO MEROZOITE SURFACE PROTEIN-1/42 MEDICAL RESEARCH COUNCIL (GB) 2004-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070003987-A1 Screening method for substance binding to merozoite surface protein-1/42 CD2BP2, MASP2, CD14 ALOX12 4520/4885CYP2A6 3890/4885TSHR 2947/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.