SCHEMBL8774333

SCHEMBL8774333

CCc1ccc(-c2cc(F)c(F)nc2F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 1/20 0.40
MAPK14 Q16539 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.36
TP53 P04637 3/20 0.35
TAAR1 Q96RJ0 1/20 0.35
LMNA P02545 2/20 0.35
METAP2 P50579 1/20 0.35
RAB9A P51151 4/20 0.35
NPC1 O15118 3/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
XDH P47989 1/20 0.34
CYP2A6 P11509 2/20 0.34
NISCH Q9Y2I1 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774763 0.98 GCGR (0.40) GCGRMAPK14SMN1; SMN2TP53TAAR1
SCHEMBL8774599 0.86 NPC1 (0.41) SMN1; SMN2TP53RAB9ANPC1NISCH
SCHEMBL8774744 0.85 GCGR (0.38) GCGRMAPK14SMN1; SMN2TP53TAAR1
SCHEMBL8774928 0.85 NPC1 (0.40) SMN1; SMN2TP53TAAR1RAB9ANPC1
SCHEMBL8774855 0.83 RARB (0.46) SMN1; SMN2TP53RAB9ANPC1NISCH
SCHEMBL8774472 0.82 RARB (0.51) MAPK14SMN1; SMN2TP53LMNARAB9A
SCHEMBL8774685 0.82 RARB (0.45) SMN1; SMN2TP53RAB9ANPC1NISCH
SCHEMBL8774890 0.81 RARB (0.50) SMN1; SMN2RAB9AGAAALDH1A1MAPT
SCHEMBL15471664 0.81 TAAR1 (0.43) GCGRMAPK14TP53TAAR1LMNA
SCHEMBL8774081 0.78 FFAR4 (0.46) SMN1; SMN2TP53LMNARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed