SCHEMBL8774928

SCHEMBL8774928

CCCc1ccc(-c2ccc(-c3cc(F)c(F)nc3F)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TP53 P04637 1/20 0.40
PKM P14618 1/20 0.40
MAPT P10636 1/20 0.39
GFER P55789 1/20 0.39
RARB P10826 3/20 0.38
MCL1 Q07820 1/20 0.38
RARA P10276 1/20 0.38
RARG P13631 1/20 0.38
NISCH Q9Y2I1 1/20 0.36
MAOB P27338 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
ALOX5 P09917 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35
HTT P42858 1/20 0.35
CYP17A1 P05093 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774599 0.98 NPC1 (0.41) NPC1RAB9ASMN1; SMN2HSD17B10TP53
SCHEMBL8774685 0.91 RARB (0.45) NPC1RAB9ASMN1; SMN2HSD17B10TP53
SCHEMBL8774890 0.89 RARB (0.50) RAB9ASMN1; SMN2HSD17B10MAPTRARB
SCHEMBL8774855 0.89 RARB (0.46) NPC1RAB9ASMN1; SMN2HSD17B10TP53
SCHEMBL8774472 0.88 RARB (0.51) RAB9ASMN1; SMN2HSD17B10TP53MAPT
SCHEMBL8774763 0.87 GCGR (0.40) NPC1RAB9ASMN1; SMN2TP53MAPT
SCHEMBL8774333 0.85 GCGR (0.40) NPC1RAB9ASMN1; SMN2TP53MAPT
SCHEMBL8774007 0.84 RAB9A (0.42) NPC1RAB9ASMN1; SMN2HSD17B10TP53
SCHEMBL8774334 0.83 NPC1 (0.40) NPC1RAB9ASMN1; SMN2HSD17B10TP53
SCHEMBL13343394 0.81 RARB (0.48) NPC1RAB9ASMN1; SMN2HSD17B10TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed