SCHEMBL8774407

SCHEMBL8774407

CCCCCC1CCC(CCc2ccc(-c3cc(F)c(F)nc3Cl)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 3/20 0.36
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C8 P10632 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
S1PR3 Q99500 1/20 0.34
RARA P10276 1/20 0.33
RARG P13631 1/20 0.33
GPR84 Q9NQS5 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
TLR8 Q9NR97 1/20 0.32
CTRC Q99895 1/20 0.32
HSD11B1 P28845 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
ITGB3 P05106 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774400 1.00 RARB (0.36) RARBGAAMAPTCYP3A4CYP2C8
SCHEMBL8775089 0.97 GPR84 (0.36) RARBGAAMAPTRARARARG
SCHEMBL8775095 0.97 GPR84 (0.36) RARBGAAMAPTRARARARG
SCHEMBL8775158 0.92 GPR84 (0.34) RARBGPR84NPC1RAB9AMAOA
SCHEMBL8775154 0.92 GPR84 (0.34) RARBGPR84NPC1RAB9AMAOA
SCHEMBL8774058 0.90 RARB (0.38) RARBGAAMAPTCYP3A4CYP2C8
SCHEMBL8774639 0.90 GPR84 (0.34) GPR84MAOAMAOBFFAR4
SCHEMBL8774053 0.90 RARB (0.38) RARBGAAMAPTCYP3A4CYP2C8
SCHEMBL8774629 0.90 GPR84 (0.34) GPR84MAOAMAOBFFAR4
SCHEMBL8775036 0.89 RARB (0.40) RARBGAAMAPTCYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed