SCHEMBL8775031

SCHEMBL8775031

CCOc1ccc(-c2ccc(C#Cc3cc(F)c(F)nc3F)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
NQO1 P15559 1/20 0.38
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 2/20 0.38
LMNA P02545 1/20 0.38
MCHR1 Q99705 1/20 0.37
XDH P47989 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
MPI P34949 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CHRNA7 P36544 1/20 0.36
MAPT P10636 1/20 0.36
ACACB O00763 7/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774805 0.96 NQO1 (0.41) CYP11B1CYP11B2NQO1ACACBSYK
SCHEMBL8774463 0.90 MCHR1 (0.41) ALDH1A1RAB9ANPC1MCHR1GAA
SCHEMBL8775170 0.90 CYP2D6 (0.46) KDM4EALDH1A1RAB9ANPC1LMNA
SCHEMBL8774435 0.85 ACACB (0.40) LMNAHSD17B10CHRNA7ACACB
SCHEMBL8774602 0.85 ACACB (0.39) KDM4EALDH1A1RAB9ALMNAHPGD
SCHEMBL8774750 0.83 FFAR1 (0.38) RAB9ANPC1GAASMN1; SMN2ACACB
SCHEMBL8774095 0.83 NR5A1 (0.41) KDM4EALDH1A1RAB9ANPC1LMNA
SCHEMBL9158464 0.82 NQO1 (0.39) CYP11B1CYP11B2NQO1KDM4EALDH1A1
SCHEMBL8774387 0.81 APP (0.46) CYP11B1CYP11B2ALDH1A1MCHR1ACACB
SCHEMBL8774994 0.81 FFAR1 (0.42) RAB9ANPC1SMN1; SMN2HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed