SCHEMBL8774867

SCHEMBL8774867

CCCCc1ccc(CCc2cc(F)c(F)nc2Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTRC Q99895 1/20 0.39
HTR2A P28223 1/20 0.37
KCNH2 Q12809 4/20 0.36
MAPT P10636 1/20 0.36
CA2 P00918 2/20 0.36
CA1 P00915 1/20 0.36
POLA1 P09884 1/20 0.36
EIF4A1 P60842 2/20 0.35
RARB P10826 2/20 0.35
RARA P10276 1/20 0.35
RARG P13631 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774859 0.96 HTR2A (0.42) HTR2AKCNH2RARBRARARARG
SCHEMBL8774238 0.91 RAB9A (0.37) MAPTCA2ALDH1A1HPGDHSD17B10
SCHEMBL8775021 0.88 TAAR1 (0.39) MAPTALDH1A1SMN1; SMN2NPC1TP53
SCHEMBL8774498 0.86 HTR2A (0.40) HTR2ACA2CA1RARBRARA
SCHEMBL8774250 0.82 RARB (0.44) CTRCMAPTEIF4A1RARBRARA
SCHEMBL8774823 0.82 HTR2A (0.46) HTR2AKCNH2RARBRARARARG
SCHEMBL8774419 0.81 RARB (0.43) CTRCMAPTEIF4A1RARBRARA
SCHEMBL8774041 0.81 HTR2A (0.49) HTR2AKCNH2RARBRARARARG
SCHEMBL8774036 0.78 RARB (0.49) HTR2AMAPTRARBRARARARG
SCHEMBL8775053 0.77 RARB (0.48) CTRCHTR2AKCNH2MAPTRARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed