SCHEMBL8774419

SCHEMBL8774419

CCCCc1ccc(-c2cc(F)c(F)nc2Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 4/20 0.43
CTRC Q99895 1/20 0.43
RARA P10276 1/20 0.40
RARG P13631 1/20 0.40
MAPT P10636 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
EIF4A1 P60842 3/20 0.39
PSMB5 P28074 1/20 0.39
MPL P40238 2/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
HSD11B1 P28845 2/20 0.38
GCGR P47871 1/20 0.38
NFKB1 P19838 1/20 0.38
MAPK1 P28482 1/20 0.38
NFKB2 Q00653 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8775053 0.96 RARB (0.48) RARBCTRCRARARARGMAPT
SCHEMBL8774679 0.94 RARB (0.50) RARBRARARARGMAPTRAB9A
SCHEMBL8774007 0.91 RAB9A (0.42) RARBCTRCRARARARGMAPT
SCHEMBL8774855 0.87 RARB (0.46) RARBCTRCRARARARGMAPT
SCHEMBL8774685 0.85 RARB (0.45) RARBCTRCRARARARGMAPT
SCHEMBL8774744 0.85 GCGR (0.38) MAPTNPC1RAB9ASMN1; SMN2TP53
SCHEMBL8775089 0.84 GPR84 (0.36) RARBCTRCRARARARGMAPT
SCHEMBL8775095 0.84 GPR84 (0.36) RARBCTRCRARARARGMAPT
SCHEMBL8774400 0.83 RARB (0.36) RARBCTRCRARARARGMAPT
SCHEMBL8774407 0.83 RARB (0.36) RARBCTRCRARARARGMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed