SCHEMBL8774498

SCHEMBL8774498

CCCCc1ccc(CCc2cc(F)c(F)nc2F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.40
CA2 P00918 2/20 0.39
CA1 P00915 1/20 0.39
RARB P10826 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HSD17B10 Q99714 2/20 0.38
HPGD P15428 1/20 0.38
RARA P10276 1/20 0.38
RARG P13631 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
TP53 P04637 2/20 0.37
NPC1 O15118 1/20 0.37
TSHR P16473 1/20 0.37
RAB9A P51151 1/20 0.37
SKP2 Q13309 1/20 0.37
GPR84 Q9NQS5 1/20 0.36
TLR8 Q9NR97 2/20 0.36
ESR1 P03372 2/20 0.36
ADRA2A P08913 2/20 0.36
ADORA3 P0DMS8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774250 0.95 RARB (0.44) RARBALDH1A1HSD17B10RARARARG
SCHEMBL8774823 0.95 HTR2A (0.46) HTR2ARARBALDH1A1HSD17B10RARA
SCHEMBL8774041 0.94 HTR2A (0.49) HTR2ARARBALDH1A1HSD17B10RARA
SCHEMBL8774036 0.91 RARB (0.49) HTR2ARARBALDH1A1HSD17B10HPGD
SCHEMBL8774829 0.90 RAB9A (0.36) CA2ALDH1A1HSD17B10SMN1; SMN2TP53
SCHEMBL8775001 0.87 PKM (0.42) RARBALDH1A1RARASMN1; SMN2LMNA
SCHEMBL8775165 0.87 TAAR1 (0.42) HTR2ATP53NPC1RAB9AGPR84
SCHEMBL8774867 0.86 CTRC (0.39) HTR2ACA2CA1RARBALDH1A1
SCHEMBL8774334 0.86 NPC1 (0.40) RARBHSD17B10RARARARGSMN1; SMN2
SCHEMBL8774813 0.84 MEN1 (0.42) ALDH1A1SMN1; SMN2LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed