SCHEMBL8774896

SCHEMBL8774896

CCc1ccc(C2CCC(CCc3cnc(Cl)c(Cl)c3)CC2)cc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.35
ESR2 Q92731 2/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
MEN1 O00255 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
SPHK1 Q9NYA1 3/20 0.33
DRD2 P14416 1/20 0.33
HRH3 Q9Y5N1 2/20 0.32
LSS P48449 1/20 0.32
MAOB P27338 1/20 0.32
KCNH2 Q12809 1/20 0.32
DGAT1 O75907 1/20 0.32
OPRL1 P41146 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774886 1.00 CYP2C9 (0.35) CYP2C9ESR2ALDH1A1LMNAMAPT
SCHEMBL8774879 0.92 MAOA (0.38) CYP2C9ESR2ALDH1A1LMNAMAPT
SCHEMBL8774872 0.92 MAOA (0.38) CYP2C9ESR2ALDH1A1LMNAMAPT
SCHEMBL8774647 0.90 SPHK1 (0.44) CYP2C9ALDH1A1LMNAMAPTMEN1
SCHEMBL8774636 0.90 SPHK1 (0.44) CYP2C9ALDH1A1LMNAMAPTMEN1
SCHEMBL8774920 0.89 SPHK1 (0.49) CYP2C9MAPTSPHK1
SCHEMBL9152491 0.84 CYP2C9 (0.40) CYP2C9ESR2ALDH1A1LMNAMAPT
SCHEMBL9152496 0.84 CYP2C9 (0.40) CYP2C9ESR2ALDH1A1LMNAMAPT
SCHEMBL8774056 0.83 DRD2 (0.38) ALDH1A1MAPTMEN1KMT2ASPHK1
SCHEMBL8774047 0.83 DRD2 (0.38) ALDH1A1MAPTMEN1KMT2ASPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed