SCHEMBL877667

SCHEMBL877667

CN(C(=O)c1ccc2c(c1)C(N1CC=CC(OC(=O)O)=C1C(F)(F)F)CC2)C1CCN(c2ccnc(N3CCCC3)n2)CC1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACACB O00763 3/20 0.32
POLB P06746 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
PDK2 Q15119 1/20 0.30
GBA1 P04062 1/20 0.30
HRH4 Q9H3N8 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30
KDM4A O75164 1/20 0.30
KDM4C Q9H3R0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878098 0.90 HRH4 (0.32) POLBHRH4HRH3KDM4AKDM4C
SCHEMBL877632 0.90 HRH4 (0.31) POLBHRH4HRH3KDM4AKDM4C
SCHEMBL877845 0.85 F10 (0.35) POLBPDK2KDM4AKDM4C
SCHEMBL878581 0.84 TLR9 (0.33) PDK2GBA1
SCHEMBL877739 0.84 KDM4A (0.31) POLBKDM4AKDM4C
SCHEMBL877666 0.77 KDM4A (0.34) ACACBPOLBADORA2AADORA1PDK2
SCHEMBL876177 0.75 F10 (0.33)
SCHEMBL877422 0.75 F10 (0.34) POLB
SCHEMBL785498 0.73 PDE4A (0.37) POLBPDK2GBA1
SCHEMBL784264 0.71 POLB (0.36) ACACBPOLBGBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed