SCHEMBL878581

SCHEMBL878581

Cc1cc(N2CCC(N(C)C(=O)c3ccc4c(c3)C(N3CC=CC(OC(=O)O)=C3C(F)(F)F)CC4)CC2)nc(N(C)C)n1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
GBA1 P04062 1/20 0.33
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
PDK2 Q15119 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL877632 0.86 HRH4 (0.31)
SCHEMBL877845 0.85 F10 (0.35) TLR9TLR8TLR7PDK2
SCHEMBL878098 0.85 HRH4 (0.32)
SCHEMBL877667 0.84 ACACB (0.32) GBA1PDK2
SCHEMBL877739 0.81 KDM4A (0.31)
SCHEMBL878580 0.77 ALDH1A1 (0.34) TLR9TLR8TLR7GBA1ALDH1A1
SCHEMBL876177 0.76 F10 (0.33)
SCHEMBL877422 0.74 F10 (0.34)
SCHEMBL785488 0.72 GBA1 (0.38) TLR9TLR8TLR7GBA1ALDH1A1
SCHEMBL878327 0.70 TLR9 (0.36) TLR9TLR8TLR7PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed