SCHEMBL877666

SCHEMBL877666

CN(C(=O)c1ccc2c(c1)C(N1C=CC=C(C(=O)O)C1C(F)(F)F)CC2)C1CCN(c2ccnc(N3CCCC3)n2)CC1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
POLB P06746 1/20 0.33
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
PDK2 Q15119 1/20 0.32
GBA1 P04062 1/20 0.32
HRH4 Q9H3N8 2/20 0.32
HRH3 Q9Y5N1 2/20 0.32
PKM P14618 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
ACACB O00763 3/20 0.31
PDE4B Q07343 1/20 0.30
SLC6A7 Q99884 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878097 0.90 KDM4A (0.35) KDM4AKDM4CPOLBPDK2HRH4
SCHEMBL877631 0.90 KDM4A (0.35) KDM4AKDM4CPOLBPDK2HRH4
SCHEMBL877844 0.84 F10 (0.37) KDM4AKDM4CPOLBPDK2
SCHEMBL878580 0.83 ALDH1A1 (0.34) KDM4AKDM4CPDK2GBA1KDM4E
SCHEMBL877667 0.77 ACACB (0.32) KDM4AKDM4CPOLBADORA2AADORA1
SCHEMBL785498 0.74 PDE4A (0.37) POLBPDK2GBA1PDE4B
SCHEMBL876176 0.73 F10 (0.32) PDK2PDE4B
SCHEMBL784264 0.73 POLB (0.36) POLBGBA1KDM4EALDH1A1LMNA
SCHEMBL877421 0.73 CCR5 (0.36) KDM4AKDM4CPOLBADORA2AADORA1
SCHEMBL784608 0.71 MEN1 (0.43) GBA1ALDH1A1PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed