SCHEMBL8776712

SCHEMBL8776712

N#Cc1cccnc1OCC(=O)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
HPGD P15428 3/20 0.53
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
CYP1A2 P05177 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
NPSR1 Q6W5P4 1/20 0.44
CTNNB1 P35222 1/20 0.43
WNT3A P56704 1/20 0.43
KDM4E B2RXH2 3/20 0.42
MAPK1 P28482 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 1/20 0.42
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.42
KMT2A Q03164 1/20 0.42
SSTR4 P31391 1/20 0.42
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15303617 0.85 KDM4E (0.50) ALDH1A1HPGDKDM4ESSTR4ALOX15
SCHEMBL3834658 0.81 KDM4E (0.44) ALDH1A1HPGDKDM4EMAPK1MEN1
SCHEMBL1280798 0.79 SSTR4 (0.43) ALDH1A1HPGDNPC1RAB9ANPSR1
SCHEMBL27712540 0.79 LMNA (0.48) ALDH1A1HPGDNPC1RAB9ACYP1A2
SCHEMBL1384171 0.79 NPC1 (0.74) ALDH1A1HPGDNPC1RAB9AL3MBTL1
SCHEMBL16794805 0.77 NPC1 (0.67) ALDH1A1HPGDNPC1RAB9ACYP1A2
SCHEMBL4034458 0.74 MAOB (0.51) NPC1RAB9AL3MBTL1MEN1KMT2A
SCHEMBL8776853 0.73 ALDH1A1 (0.64) ALDH1A1HPGDNPC1RAB9ACYP1A2
SCHEMBL21748902 0.73 SSTR4 (0.59) ALDH1A1CYP2C9KDM4ESSTR4
SCHEMBL8776818 0.72 CYP11B1 (0.48) ALDH1A1HPGDNPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed