SCHEMBL8776770

SCHEMBL8776770

CCS(=O)(=O)c1ccc(-c2cc(C#N)c(OC)nc2-c2cccc(F)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 8/20 0.45
CNR1 P21554 5/20 0.43
CNR2 P34972 1/20 0.43
SQOR Q9Y6N5 3/20 0.40
AKT1 P31749 1/20 0.40
AKT2 P31751 1/20 0.40
FLT1 P17948 1/20 0.40
FLT4 P35916 1/20 0.40
KDR P35968 1/20 0.40
KDM4E B2RXH2 2/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8093568 0.90 PTGS2 (0.46) SCN9ACNR1CNR2SQOR
SCHEMBL8776720 0.90 PTGS2 (0.47) SCN9ACNR1CNR2SQORKDM4E
SCHEMBL8086726 0.89 CA4 (0.46) SCN9ACNR1CNR2SQORKDM4E
SCHEMBL8776752 0.88 CNR1 (0.48) SCN9ACNR1CNR2SQORAKT1
SCHEMBL8776866 0.85 KDM4E (0.43) CNR1CNR2AKT1AKT2KDM4E
SCHEMBL8776778 0.83 CNR1 (0.41) CNR1CNR2SQORAKT1AKT2
SCHEMBL8776740 0.81 CNR1 (0.52) CNR1CNR2
SCHEMBL8776745 0.80 KDM4E (0.46) CNR1AKT1AKT2KDM4EPOLB
SCHEMBL215205 0.79 PTGS2 (0.53) CNR1CNR2SQOR
SCHEMBL8093195 0.78 PTGS2 (0.47) CNR1CNR2SQORKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP claimed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO claimed