SCHEMBL8776866

SCHEMBL8776866

CCS(=O)(=O)c1ccc(-c2cc(C#N)c(OC)nc2-c2ccc(C)c(C)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.43
POLB P06746 2/20 0.43
CNR1 P21554 8/20 0.40
MEN1 O00255 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KMT2A Q03164 2/20 0.40
HPGD P15428 1/20 0.40
CNR2 P34972 4/20 0.39
AKT1 P31749 1/20 0.38
AKT2 P31751 1/20 0.38
RORC P51449 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GAA P10253 1/20 0.36
PTGS2 P35354 1/20 0.34
CTSK P43235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8087289 0.89 PTGS2 (0.46) KDM4EPOLBCNR1MEN1ALDH1A1
SCHEMBL8096123 0.88 PTGS2 (0.47) KDM4EPOLBCNR1MEN1ALDH1A1
SCHEMBL8776720 0.86 PTGS2 (0.47) KDM4EPOLBCNR1MEN1KMT2A
SCHEMBL8776752 0.85 CNR1 (0.48) CNR1CNR2AKT1AKT2RORC
SCHEMBL8776770 0.85 SCN9A (0.45) KDM4EPOLBCNR1CNR2AKT1
SCHEMBL8776778 0.83 CNR1 (0.41) KDM4EPOLBCNR1CNR2AKT1
SCHEMBL8776745 0.83 KDM4E (0.46) KDM4EPOLBCNR1ALDH1A1HPGD
SCHEMBL8776740 0.81 CNR1 (0.52) CNR1CNR2
SCHEMBL8776824 0.81 CNR1 (0.63) CNR1CNR2
SCHEMBL8087140 0.80 KDM4E (0.43) KDM4EPOLBCNR1MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP claimed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO claimed