SCHEMBL8776897

SCHEMBL8776897

COc1ccc([C@]2(C)O[C@H]2C(=O)O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.44
CA1 P00915 3/20 0.43
CA2 P00918 3/20 0.43
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
EDNRA P25101 2/20 0.40
EDNRB P24530 1/20 0.40
CHRNA1 P02708 1/20 0.39
CHRNG P07510 1/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9750487 1.00 HSD11B1 (0.44) HSD11B1CA1CA2ATML3MBTL1
SCHEMBL9692259 0.85 ATM (0.50) HSD11B1CA1CA2ATML3MBTL1
SCHEMBL9750499 0.84 HCAR2 (0.50) CES2CES1KMT2ANPC1MAPT
SCHEMBL16108980 0.83 GAA (0.43) HSD11B1CA1CA2ATML3MBTL1
SCHEMBL2234611 0.80 CRHBP (0.44) HSD11B1KMT2AMAPTMAPK1CHRNB2
SCHEMBL18316474 0.80 CRHBP (0.44) HSD11B1KMT2AMAPTMAPK1CHRNB2
SCHEMBL31354802 0.80 CRHBP (0.44) HSD11B1KMT2AMAPTMAPK1CHRNB2
SCHEMBL16109494 0.80 ATM (0.40) HSD11B1CA1CA2ATML3MBTL1
SCHEMBL16109050 0.80 ALDH1A1 (0.46) ATML3MBTL1KMT2ANPC1MAPT
SCHEMBL16108652 0.80 HPGD (0.43) HSD11B1CA1CA2ATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0453330-B2 Process for the preparation of (-) (2R,3S)-2,3-epoxy-3-(4-methoxyphenyl) propionic acid methylester and its enantiomer SYNTHELABO (FR) 1997-12-03 EP claimed
JP-2145564-A None JP disclosed
JP-4217969-A None JP disclosed
US-RE34935-E Method for preparing (+)-(2S,3S)-3-hydroxy-2-(4-methoxyphenyl)-2,3-dihydro-5H-1,5-benzothiazepine-4-one and chlorinated derivatives thereof SYNTHELABO (FR) 1995-05-09 US disclosed
JP-H04217969-A PREPARATION OF (-)-(METHYL-(2R,3S)-2,3-EPOXY-3-(4-METHOXYPHENYL)PROPIONATE) AND ENANTIOMER THEREOF SYNTHELABO SA 1992-08-07 JP disclosed
JP-H02145564-A PREPARATION OF PROPIONIC ACID DERIVATIVE SYNTHELABO SA 1990-06-05 JP disclosed