SCHEMBL8779221

SCHEMBL8779221

C[C@H](N)C(=O)NC(=O)Oc1nccc(OCC(F)(F)C(F)F)c1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.38
KMT2A Q03164 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 5/20 0.34
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 2/20 0.34
CARM1 Q86X55 2/20 0.34
PRMT6 Q96LA8 2/20 0.34
LMNA P02545 2/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
PAX8 Q06710 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
AAK1 Q2M2I8 6/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GSK3B P49841 2/20 0.32
MAPK1 P28482 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779232 0.90 GSK3B (0.39) MAPTCARM1PRMT6AAK1CYP2C9
SCHEMBL8779252 0.88 CARM1 (0.34) MAPTCARM1PRMT6AAK1GSK3B
SCHEMBL8779141 0.87 AAK1 (0.33) MAPTCARM1PRMT6AAK1GSK3B
SCHEMBL9233029 0.85 KMT2A (0.41) HTTKMT2ASMN1; SMN2MAPTKDM4E
SCHEMBL8779212 0.83 HPGD (0.38) KMT2ASMN1; SMN2KDM4ECARM1PRMT6
SCHEMBL8779176 0.83 HPGD (0.38) KMT2ASMN1; SMN2KDM4ECARM1PRMT6
SCHEMBL8883898 0.83 KMT2A (0.39) HTTKMT2ASMN1; SMN2MAPTKDM4E
SCHEMBL8779292 0.82 CARM1 (0.35) SMN1; SMN2CARM1PRMT6AAK1CYP3A4
SCHEMBL8779316 0.82 MME (0.39)
SCHEMBL8779136 0.81 IKBKB (0.37) SMN1; SMN2MAPTKDM4ECARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed