SCHEMBL8779241

SCHEMBL8779241

CCCCCOc1ccnc(OC(=O)NC(=O)CN)c1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.40
NPC1 O15118 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
MEN1 O00255 1/20 0.37
NR1I2 O75469 1/20 0.37
CHRM2 P08172 1/20 0.37
ADRA2A P08913 1/20 0.37
MAPT P10636 1/20 0.37
OPRK1 P41145 1/20 0.37
HTR2B P41595 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779257 0.99 LMNA (0.41) LMNANPC1CYP3A4CYP1A2CYP2D6
SCHEMBL8779138 0.96 SMN1; SMN2 (0.39) LMNANPC1CYP3A4CYP1A2CYP2D6
SCHEMBL8779273 0.93 IKBKB (0.38) LMNANPC1CYP3A4CYP1A2CYP2D6
SCHEMBL8779277 0.89 SMN1; SMN2 (0.35) LMNASMN1; SMN2KMT2A
SCHEMBL8779087 0.88 IKBKB (0.34) LMNASMN1; SMN2MEN1KMT2A
SCHEMBL8779326 0.88 SMN1; SMN2 (0.39) LMNASMN1; SMN2KMT2A
SCHEMBL8786169 0.85 LMNA (0.40) LMNANPC1CYP3A4CYP1A2CYP2D6
SCHEMBL8779253 0.85 HTT (0.39) HDAC6
SCHEMBL8779165 0.84 XIAP (0.38) LMNANPC1CYP3A4CYP1A2CYP2D6
SCHEMBL8785900 0.84 LMNA (0.45) LMNANPC1CYP3A4SMN1; SMN2NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed