SCHEMBL8779273

SCHEMBL8779273

CCCOc1ccnc(OC(=O)NC(=O)CN)c1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.38
MAPT P10636 3/20 0.35
HSD17B10 Q99714 1/20 0.35
LMNA P02545 4/20 0.33
HPGD P15428 1/20 0.33
PLK1 P53350 1/20 0.33
CARM1 Q86X55 1/20 0.32
ATM Q13315 1/20 0.32
TSHR P16473 1/20 0.32
CCNT1 O60563 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CDK9 P50750 1/20 0.32
CCNA1 P78396 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
HTT P42858 2/20 0.32
GRM5 P41594 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779138 0.94 SMN1; SMN2 (0.39) MAPTHSD17B10LMNAHPGDSMN1; SMN2
SCHEMBL8779241 0.93 LMNA (0.40) MAPTLMNASMN1; SMN2CYP2C19FAAH
SCHEMBL8779257 0.92 LMNA (0.41) MAPTLMNASMN1; SMN2CYP2C19FAAH
SCHEMBL8779326 0.90 SMN1; SMN2 (0.39) IKBKBLMNAHPGDCARM1GRM5
SCHEMBL8779277 0.89 SMN1; SMN2 (0.35) LMNACARM1SMN1; SMN2ALDH1A1
SCHEMBL8779087 0.88 IKBKB (0.34) IKBKBLMNAHPGDCARM1SMN1; SMN2
SCHEMBL8779253 0.87 HTT (0.39) HTTGAAACACB
SCHEMBL8779250 0.86 MEN1 (0.42) MAPTLMNAHPGDTSHRSMN1; SMN2
SCHEMBL8779284 0.85 NFKB1 (0.32) CARM1
SCHEMBL8779122 0.84 MAPT (0.33) MAPTHPGDCARM1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed